5-Iodoresiniferatoxin [535974-91-5]

MedChem Express

5-Iodoresiniferatoxin [535974-91-5]

14

535974-91-5

Research Use Only

C37H39IO9

754.60

5-Iodoresiniferatoxin (I-RTX) is a selective TRPV1 antagonist, with an IC50s of 0.7 and 5.4 nM for rat and human receptors, respectively. 5-Iodoresiniferatoxin induces TRPV1-dependent hypothermia in vivo[1].

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