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A-81282

HY-101823A
MedChem Express
Molecular Weight429.47
Product group Chemicals
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Overview

  • Supplier
    MedChem Express
  • Product Name
    A-81282
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Molecular Formula
    C23H23N7O2
  • Molecular Weight
    429.47
  • Scientific Description
    A-81282 (Abbott 81282) is an antagonist of angiotensin IIs AT1 receptor, with a p A2 value of 9.64 at the AT1 receptor in rabbit aorta. A-81282 also demonstrates significant inhibitory action on the binding of [125i]_Sar1_lle8_Angiotensin_ll to rat liver membranes, with a p KI value of 8.505. A-81282 has antihypertensive activity and can effectively lower blood pressure in renal artery-ligated rats [1] .
  • SMILES
    O=C(C1=CN=CN=C1N(CCCC)CC2=CC=C(C3=CC=CC=C3C4=NN=NN4)C=C2)O
  • UNSPSC
    12352200