AM251
ORB341682
CAS Number183232-66-8
Product group Chemicals
Molecular Weight555.2388
Overview
- SupplierBiorbyt
- Product NameAM251 [183232-66-8]
- Delivery Days Customer16
- CAS Number183232-66-8
- CertificationResearch Use Only
- Molecular FormulaC22H21CL2IN4O
- Molecular Weight555.2388
- Scientific DescriptionAM251 is a potent CB1 receptor antagonist (IC50 = 8 nM, Ki = 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also potent GPR55 agonist (EC50 = 39 nM).
- SMILESIC1=CC=C(C=C1)C2N(N=C(C(=O)NN3CCCCC3)C=2C)C4=C(Cl)C=C(Cl)C=C4
- UNSPSC12352200