AR-C 118925XX
M6457
CAS Number216657-60-2
Product group Chemicals
Molecular Weight537.59
Overview
- SupplierAbMole BioScience
- Product NameAR-C 118925XX
- Delivery Days Customer9
- CAS Number216657-60-2
- Category SupplierChemical
- CertificationResearch Use Only
- Molecular FormulaC28H23N7O3S
- Molecular Weight537.59
- Scientific DescriptionAR-C 118925XX is a selective, competitive P2Y2 receptor antagonist. AR-C 118925XX is inactive against a panel of 37 other receptors at a concentration of 10 uM. AR-C 118925XX inhibits ATP-gammaS-induced mucin secretion in bronchial epithelial cells (IC50 = 1 uM). AR-C 118925XX inhibits P2Y2 receptor-induced bèta-arrestin translocation in vitro (pA2 = 37.2-51.3 nM).
- UNSPSC12352200