Asenapine-13C,d3

MedChem Express

Asenapine-13C,d3

5

C20 13CH17D3ClNO5

405.85

Asenapine- 13 C,d 3 is 13 C and deuterated labeled Asenapine (HY-10121). Asenapine (Org 5222), an atypical antipsychotic, is an antagonist of serotonin receptors ( pK i : 8.4-10.5), adrenoceptors ( pK i : 8.9-9.5), dopamine receptors ( pK i : 8.9-9.4) and histamine receptors ( pK i : 8.2-9.0). Asenapine can be used in the research of schizophrenia and bipolar disorder [1] [2] .

ClC1=CC(C2C(CN(C2)[13C]([2H])([2H])[2H])C3=C4C=CC=C3)=C(O4)C=C1.O=C(O)/C=C\C(O)=O

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