beta2AR/M-receptor agonist-1 [2230520-62-2]

TargetMol Chemicals

beta2AR/M-receptor agonist-1 [2230520-62-2]

999

Chemical

Research Use Only

bèta2AR/M-receptor agonist-1

C43H56BrN3O7

806.82

beta2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and beta2 adrenoceptor agonist (MABA), exhibits dual potency towards beta2 adrenoceptor and muscarinic receptor, with an EC50 value of 9.2 nM for beta2 adrenoceptor and a Ki value of 30.2 nM for the muscarinic receptor, and an EC50 value of 4.0 nM highlighting its MABA activity [1].

3 years

[Br-].O[C@H](CNCCCOc1ccc(OCCC[N+]23CCC(CC2)[C@@H](C3)OC[C@@](O)(C2CCCC2)c2ccccc2)cc1)c1ccc(O)c2[nH]c(=O)ccc12

-20°C

51202000