BI-4924

Biorbyt

BI-4924 [2244452-09-1]

10

2244452-09-1

Research Use Only

C21H20CL2N2O6S

499.3643

BI-4924 (BI 4924) is a potent, selective NADH/NAD+-competitive PHGDH inhibitor with IC50 of 2 nM.BI-4924 splays high selectivity against the majority of other dehydrogenase targets.

ClC1=C(C(C([H])([H])[H])=C([H])C2=C1C([H])=C(C(N([H])[C@]([H])(C([H])([H])O[H])C1C([H])=C([H])C(=C([H])C=1[H])S(C([H])([H])C(=O)O[H])(=O)=O)=O)N2C([H])([H])[H])Cl

12352200