BIP-135
M8272
CAS Number941575-71-9
Product group Chemicals
Molecular Weight421.24
Overview
- SupplierAbMole BioScience
- Product NameBIP-135
- Delivery Days Customer9
- CAS Number941575-71-9
- Category SupplierChemical
- CertificationResearch Use Only
- Molecular FormulaC21H13BrN2O3
- Molecular Weight421.24
- Scientific DescriptionBIP-135 is a potent inhibitor of glycogen synthase kinase-3 (GSK3) found to be relatively selective for GSK-3bèta (21 nM) over GSK-3alfa with modest activity toward PKCbèta (bèta1: 980 nM; bèta2: 219 nM), DYRK1B (590 nM), and PI3Kalfa (870 nM).
- UNSPSC12352200