Bio-Connect

BMS-1166-N-piperidine-CO-N-piperazine (dihydrochloride) [2691796-83-3]

HY-131386A
MedChem Express
Product group Molecular Biology
Sign in to order and to see your custom pricing.
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    MedChem Express
  • Product Name
    BMS-1166-N-piperidine-CO-N-piperazine (dihydrochloride) [2691796-83-3]
  • Delivery Days Customer
    10
  • CAS Number
    2691796-83-3
  • Certification
    Research Use Only
  • Estimated Purity
    95.01
  • Molecular Formula
    C41H45Cl3N4O5
  • Molecular Weight
    780.18
  • Scientific Description
    BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride incorporates a ligand for PD-1/PD-L1 immune checkpoint, and a PROTAC linker. BMS-1166-N-piperidine-CO-N-piperazine dihydrochloride can be used in the synthesis of PROTAC PD-1/PD-L1 degrader-1 (HY-131183). PROTAC PD-1/PD-L1 degrader-1 inhibits PD-1/PD-L1 interaction with an IC50 of 39.2 nM[1].
  • SMILES
    N#CC1=CC=CC(COC2=CC(OCC3=CC=CC(C4=CC=C5OCCOC5=C4)=C3C)=C(C=C2CN6CCCCC6C(N7CCNCC7)=O)Cl)=C1.Cl.Cl
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    41115800