BRD-IN-3
T10604
Overview
- SupplierTargetMol Chemicals
- Product NameBRD-IN-3
- Delivery Days Customer79
- CAS Number2351938-32-2
- Category SupplierChemical
- Chemical NameBRD-IN-3
- Molecular FormulaC21H25N5O3
- Molecular Weight395.45
- Scientific DescriptionBRD-IN-3 is a highly potent PCAF bromodomain (BRD) inhibitor (IC50: 7 nM). It also exhibits activity against GCN5 and FALZ.
- Shelf life instruction3 years
- SMILESN([C@@H]1C[C@@H](CN(C)C1)C=2C=C3C(=CC2)OCCO3)C4=NC5=C(C(=O)N4C)NC=C5
- Storage Instruction-20°
- UNSPSC12352200
References
- Huang L, et al. Discovery of Pyrrolo[3,2- d]pyrimidin-4-one Derivatives as a New Class of Potent and Cell-Active Inhibitors of P300/CBP-Associated Factor Bromodomain. J Med Chem. 2019 May 9;62(9):4526-4542.Read more