Brompheniramine (maleate) (Standard)

MedChem Express

Brompheniramine (maleate) (Standard) [980-71-2]

9

Research Use Only

Brompheniramine (maleate) (Standard) is the analytical standard of Brompheniramine (maleate). This product is intended for research and analytical applications. Brompheniramine ((+/-)-Brompheniramine) maleate is a potent and orally active antihistamine of the alkylamine class. Brompheniramine maleate is a selective histamine H1 receptor antagonist with a Kd of 6.06 nM. Brompheniramine maleate can block the hERG channels, calcium channels, and sodium channels with IC 50 s of 0.90 microM, 16.12 microM and 21.26 microM, respectively. Brompheniramine maleate has anticholinergic, antidepressant and anesthetic properties and can be used for allergic rhinitis research [1] [2] [3] [4] .

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