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Buparlisib (BKM120)

S2247
Selleck Chemicals
Estimated Purity...
Product group Chemicals
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Overview

  • Supplier
    Selleck Chemicals
  • Product Name
    Buparlisib (BKM120) [944396-07-0]
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Estimated Purity
    ...
  • Scientific Description
    Buparlisib (BKM120, NVP-BKM120) is a selective PI3K inhibitor of p110alpha/beta/delta/gamma with IC50 of 52 nM/166 nM/116 nM/262 nM in cell-free assays, respectively. Reduced potency against VPS34, mTOR, DNAPK, with little activity to PI4Kbeta. Buparlisib induces apoptosis. Phase 2.
  • Storage Instruction
    -80°C
  • UNSPSC
    51202000

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