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CBP/p300-IN-8

T39826
TargetMol Chemicals
CAS Number2304416-91-7
Product group Chemicals
Molecular Weight461.562
Price on request
Packing Size
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    CBP/p300-IN-8
  • Delivery Days Customer
    1001
  • CAS Number
    2304416-91-7
  • Category Supplier
    Chemical
  • Chemical Name
    CBP/p300-IN-8
  • Molecular Formula
    C27H31N3O4
  • Molecular Weight
    461.562
  • Scientific Description
    CBP/p300-IN-8 is a potent inhibitor of the CBP/P300 family of bromodomains . CBP/p300-IN-8 inhibits CBP ( IC 50 =0.01-0.1 uΜ) and BRD4 ( IC 50 =1-1000 uΜ) activity.
  • Shelf life instruction
    3 years
  • SMILES
    COC(=O)N1[C@@H](C)CCc2c1ccc1n([C@H]3CCC[C@@H](C3)C(O)=O)c(Cc3ccccc3)nc21
  • Storage Instruction
    -20°
  • UNSPSC
    12352200

References

  • Shawn E.R. Schiller, et al. Tetrahydro-imidazo quinoline compositions as cbp/p300 inhibitors. WO2019055877A1.