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CCG258208

HY-109562
MedChem Express
CAS Number2055990-90-2
Product group Chemicals
Molecular Weight452.48
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Overview

  • Supplier
    MedChem Express
  • Product Name
    CCG258208 [2055990-90-2]
  • Delivery Days Customer
    10
  • CAS Number
    2055990-90-2
  • Certification
    Research Use Only
  • Molecular Formula
    C24H25FN4O4
  • Molecular Weight
    452.48
  • Scientific Description
    CCG258208 (GRK2-IN-1) is a potent and selective GRK2 ( G protein-coupled receptor kinase 2 ) inhibitor ( IC 50 =30 nM) while maintaining 230-fold selectivity over GRK5 ( IC 50 =7.09 microM) and more than 2500-fold selectivity over GRK1 ( IC 50 =87.3 microM), PKA, and ROCK1. CCG258208 can be used in heart failure research [1] .
  • SMILES
    FC1=C(C(NCC2=NNC=C2)=O)C=C([C@H]3[C@H](COC4=CC=C(OCO5)C5=C4)CNCC3)C=C1
  • UNSPSC
    12352200