CGP 20712

MedChem Express

CGP 20712

5

Research Use Only

C23H25F3N4O5

494.46

CGP 20712 is a highly selective beta1-adrenoceptor antagonist ( K i =0.3 nmol/L). CGP 20712s primary mechanism of action is through competitively binding to beta1-receptors, thereby blocking the positive chronotropic effects of adrenaline and noradrenaline [1] .

O=C(N)C1=CC(OCCNCC(O)COC2=CC=C(C3=NC(C(F)(F)F)=CN3C)C=C2)=CC=C1O

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