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CK2/ERK8-IN-1

Research Use Only
HY-135906
MedChem Express
CAS Number1085822-09-8
DownloadMSDS
Product group Chemicals
Estimated Purity99.0
Molecular Weight534.82
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Overview

  • Supplier
    MedChem Express
  • Product Name
    CK2/ERK8-IN-1 [1085822-09-8]
  • Delivery Days Customer
    9
  • CAS Number
    1085822-09-8
  • Certification
    Research Use Only
  • Estimated Purity
    99.0
  • Molecular Formula
    C11H9Br4N3O2
  • Molecular Weight
    534.82
  • Scientific Description
    CK2/ERK8-IN-1 is a dual casein kinase 2 (CK2) (Ki of 0.25 microM) and ERK8 (MAPK15, ERK7) inhibitor with IC50s of 0.50 microM. CK2/ERK8-IN-1 also binds to PIM1, HIPK2 (homeodomain-interacting protein kinase 2), and DYRK1A with Kis of 8.65 microM, 15.25 microM, and 11.9 microM, respectively. CK2/ERK8-IN-1 has pro-apoptotic efficacy[1].
  • SMILES
    O=C(O)CN1C2=C(Br)C(Br)=C(Br)C(Br)=C2N=C1N(C)C
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200