Delequamine

MedChem Express

Delequamine

5

Research Use Only

C18H26N2O3S

350.48

Delequamine (RS-15385-197) is an orally active and selective alpha2-adrenergic receptor antagonist with a pK i of 9.5 for alpha2-adrenoceptors in rat cortex. Delequamine shows >1000 fold selectivity against 5-HT1A receptors and alpha1-adrenoceptors. Delequamine can be used for the study of erectile dysfunction [1] .

CS(=O)(N1[C@@]2([H])C[C@@]3([H])C4=CC=C(OC)C=C4CCN3C[C@@]2([H])CCC1)=O

12352200