Desmethyl cariprazine

MedChem Express

Desmethyl cariprazine [839712-15-1]

10

839712-15-1

98.06

C20H30Cl2N4O

413.38

Desmethyl cariprazine is an active metabolite of Cariprazine [1] . Cariprazine, an antipsychotic agent candidate, exhibits high affinity for the D3 (K i =0.085 nM) and D2 (0.49 nM) receptors, and moderate affinity for the 5-HT1A receptor (2.6 nM) [2] .

O=C(NC)N[C@@H]1CC[C@@H](CCN2CCN(C3=CC=CC(Cl)=C3Cl)CC2)CC1

-20°C,2°C to 8°C

12352200