DYRK1-IN-1 [2814486-79-6]

TargetMol Chemicals

DYRK1-IN-1 [2814486-79-6]

10

Chemical

Research Use Only

DYRK1-IN-1

C12H12N6

240.26

DYRK1-IN-1 is a highly selective and ligand-efficient DYRK1A inhibitor that inhibits DYRK1A phosphorylation activity with an IC50 value of 220 nM. It exhibits good permeability and cellular activity without P-glycoprotein liability, making it suitable for research on central nervous system penetrant DYRK1A chemical probes [1].

3 years

N(C)(C)C=1N=C(C2=C3N(N=C2)N=CC=C3)C=CN1

-20°C

51202000