Elenestinib

MedChem Express

Elenestinib

10

Research Use Only

98.82

C27H29FN10O

528.58

Elenestinib (BLU-263) is a potent and orally active tyrosine kinase inhibitor that has minimal brain penetration. Elenestinib inhibits KIT D816V with an IC50 value of 0.2 nM. MElenestinib has the potential for the research of systemic mastocytosis (SM)[1][2][3].

OCCN1C=C(C=N1)C2=CN3N=CN=C(N4CCN(C5=NC=C([C@@](N)(C6=CC=C(C=C6)F)C)C=N5)CC4)C3=C2

-20°C

12352200