Ep300/CREBBP-IN-2 [2259641-59-1]

TargetMol Chemicals

Ep300/CREBBP-IN-2 [2259641-59-1]

999

Chemical

Research Use Only

Ep300/CREBBP-IN-2

C26H27F3N4O4

516.51

Ep300/CREBBP-IN-2 (Example 73) is a potent, orally bioavailable inhibitor of Ep300 and CREBBP, with IC50 values of 0.052 microM and 0.148 microM, respectively, and is used in cancer research [1].

3 years

COc1ccc(cc1)C1(CCC(F)(F)CC1)C(=O)N1C[C@H](F)C[C@@H]1C(=O)Nc1ccc2NC(=O)Cc2n1

-20°C

51202000