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EP4 receptor antagonist 1 [2287259-07-6]

EP4 receptor antagonist 1 [2287259-07-6]

T11211
TargetMol Chemicals
CAS Number2287259-07-6
Product group Chemicals
Estimated Purity99.53%
Molecular Weight458.43
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    EP4 receptor antagonist 1
  • Delivery Days Customer
    9
  • CAS Number
    2287259-07-6
  • Category Supplier
    Chemical
  • Certification
    Research Use Only
  • Chemical Name
    EP4 receptor antagonist 1
  • Estimated Purity
    99.53%
  • Molecular Formula
    C23H21F3N4O3
  • Molecular Weight
    458.43
  • Scientific Description
    EP4 Receptor Antagonist 1 is a highly potent and selective competitive prostanoid EP4 receptor antagonist, effective for cancer immunotherapy. It inhibits both human and mouse EP4 receptors with IC50 values of 6.1 nM and 16.2 nM, respectively, while displaying minimal activity (IC50s >10 microM) against human EP1, EP2, and EP3 receptors.
  • Shelf life instruction
    3 years
  • SMILES
    C\C=C\c1nnn(Cc2ccc(cc2)C(F)(F)F)c1C(=O)N[C@@H](C)c1ccc(cc1)C(O)=O
  • Storage Instruction
    -20°C
  • UNSPSC
    51202000