EPI-001 (Standard) [227947-06-0]

HY-100348R
Product group Assays
Overview
- SupplierMedChem Express
- Product NameEPI-001 (Standard) [227947-06-0]
- Delivery Days Customer5
- CAS Number227947-06-0
- CertificationResearch Use Only
- Molecular FormulaC21H27ClO5
- Molecular Weight394.89
- Scientific DescriptionEPI-001 (Standard) is the analytical standard of EPI-001. This product is intended for research and analytical applications. EPI-001, a selective inhibitor of Androgen Receptor (AR), targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC50 of ~6 microM. EPI-001 is also a selective modulator of PPARgamma. EPI-001 is active against castration-resistant prostate cancer[1][2][3].
- SMILESOCC(O)COC1=CC=C(C(C)(C2=CC=C(OCC(O)CCl)C=C2)C)C=C1
- UNSPSC41116135