Bio-Connect

EPI-001 (Standard) [227947-06-0]

Research Use Only
HY-100348R
MedChem Express
Product group Assays
Sign in to order and to see your custom pricing.
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    MedChem Express
  • Product Name
    EPI-001 (Standard) [227947-06-0]
  • Delivery Days Customer
    5
  • CAS Number
    227947-06-0
  • Certification
    Research Use Only
  • Molecular Formula
    C21H27ClO5
  • Molecular Weight
    394.89
  • Scientific Description
    EPI-001 (Standard) is the analytical standard of EPI-001. This product is intended for research and analytical applications. EPI-001, a selective inhibitor of Androgen Receptor (AR), targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC50 of ~6 microM. EPI-001 is also a selective modulator of PPARgamma. EPI-001 is active against castration-resistant prostate cancer[1][2][3].
  • SMILES
    OCC(O)COC1=CC=C(C(C)(C2=CC=C(OCC(O)CCl)C=C2)C)C=C1
  • UNSPSC
    41116135