EPI-001 (Standard)

MedChem Express

EPI-001 (Standard) [227947-06-0]

5

Research Use Only

EPI-001 (Standard) is the analytical standard of EPI-001. This product is intended for research and analytical applications. EPI-001, a selective inhibitor of Androgen Receptor (AR) , targets transactivation unit 5 (Tau-5) of the AR. EPI-001 can inhibit transactivation of the AR amino-terminal domain (NTD), with an IC 50 of ~6 microM. EPI-001 is also a selective modulator of PPARgamma . EPI-001 is active against castration-resistant prostate cancer [1] [2] [3] .

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