Eplivanserin (hemifumarate)

MedChem Express

Eplivanserin (hemifumarate) [130580-02-8]

10

130580-02-8

Research Use Only

98.07

C19H21FN2O2.1/2C4H4O4

386.43

Eplivanserin (SR-46349) hemifumarate is a potent, selective and orally active 5-HT 2A receptor antagonist, with an IC 50 of 5.8 nM in rat cortical membrane, and a K d of 1.14 nM. Eplivanserin hemifumarate displays >20-fold selectivity more selective for 5-HT 2A than 5-HT 2B and 5-HT 2C [1] [2] .

O=C(O)/C=C/C(O)=O.OC(C=C1)=CC=C1/C=C/C(C2=C(C=CC=C2)F)=N/OCCN(C)C.[1/2]

2°C to 8°C

12352200