Estrogen receptor modulator 8 [2170766-56-8]

TargetMol Chemicals

Estrogen receptor modulator 8 [2170766-56-8]

16

Chemical

Research Use Only

Estrogen receptor modulator 8

C25H24F4N2O2

460.46

Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR alpha with potent efficacy (IC50 = 0.437 nM in MCF-7 cells) and effectively hampers MCF-7 cell proliferation (IC50 = 0.1 nM) [1].

3 years

C(C(C)(C)F)N1[C@@H](C2=C(C=3C(N2)=CC=CC3F)C[C@H]1C)C4=C(F)C=C(/C=C/C(O)=O)C=C4F

-20°C

51202000