Bio-Connect

(E/Z)-GSK5182

HY-111226A
MedChem Express
Estimated Purity99.17
Product group Chemicals
Molecular Weight417.54
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Overview

  • Supplier
    MedChem Express
  • Product Name
    (E/Z)-GSK5182
  • Delivery Days Customer
    9
  • Certification
    Research Use Only
  • Estimated Purity
    99.17
  • Molecular Formula
    C27H31NO3
  • Molecular Weight
    417.54
  • Scientific Description
    (E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor gamma (ERRgamma) with an IC 50 of 79 nM [1] . GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma [1] [2] [3] .
  • SMILES
    OCCC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)OCCN(C)C)\C3=CC=C(C=C3)O
  • Storage Instruction
    -20°C,2°C to 8°C
  • UNSPSC
    12352200