(E/Z)-GSK5182
HY-111226A
Overview
- SupplierMedChem Express
- Product Name(E/Z)-GSK5182
- Delivery Days Customer9
- CertificationResearch Use Only
- Estimated Purity99.17
- Molecular FormulaC27H31NO3
- Molecular Weight417.54
- Scientific Description(E/Z)-GSK5182 is a racemic compound of (E)-GSK5182 and (Z)-GSK5182 isomers. GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor gamma (ERRgamma) with an IC 50 of 79 nM [1] . GSK5182 also induces reactive oxyen species (ROS) generation in hepatocellular carcinoma [1] [2] [3] .
- SMILESOCCC/C(C1=CC=CC=C1)=C(C2=CC=C(C=C2)OCCN(C)C)\C3=CC=C(C=C3)O
- Storage Instruction-20°C,2°C to 8°C
- UNSPSC12352200