FR139317

MedChem Express

FR139317 [142375-60-8]

5

142375-60-8

Research Use Only

C33H44N6O5

604.74

FR139317 (PD 147953) is a selective ET A receptor antagonist. FR139317 inhibits cerebral activation by intraventricular endothelin-1 in conscious rats. FR139317 also ameliorates cerebral vasospasm in dogs [1] [2] .

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