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FT001 [1778655-51-8]
T27392
Overview
- SupplierTargetMol Chemicals
- Product NameFT001 [1778655-51-8]
- Delivery Days Customer9
- Category SupplierChemical
- CertificationResearch Use Only
- Chemical NameFT001
- Molecular FormulaC25H29N3O4S
- Molecular Weight467.58
- Scientific DescriptionFT001 is a potent, selective and orally available inhibitor of BET Bromodomain with antitumor activity. FT001 inhibited the expression of MYC with the IC50 value of 0.46 microM). FT001 has potent antiproliferative effects against MV-4-11 and demonstrates significant MYC mRNA suppression both in vitro and in vivo.
- Shelf life instruction3 years
- SMILESC(=O)(N1C=2C(N(C(C)=O)[C@@H](C)C1)=CC=C(C2)C3=CC=C(C=C3)N4CCS(=O)(=O)CC4)C5CC5
- Storage Instruction-20°C
- UNSPSC12352200
References
- Millan DS, et al. Design and Optimization of Benzopiperazines as Potent Inhibitors of BET Bromodomains. ACS Med Chem Lett. 2017 Jul 14;8(8):847-852.Read more