Bio-Connect
CgoaEGY7ReSEdfx6AAAAAO_pso0814.png
CgoaEGY7ReSEdfx6AAAAAO_pso0814.png
CgoaEGY7ReSEdfx6AAAAAO_pso0814.png

FT001 [1778655-51-8]

Research Use Only
T27392
TargetMol Chemicals
Molecular Weight467.58
Product group Chemicals
Price on request
Packing Size
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    FT001 [1778655-51-8]
  • Delivery Days Customer
    9
  • Category Supplier
    Chemical
  • Certification
    Research Use Only
  • Chemical Name
    FT001
  • Molecular Formula
    C25H29N3O4S
  • Molecular Weight
    467.58
  • Scientific Description
    FT001 is a potent, selective and orally available inhibitor of BET Bromodomain with antitumor activity. FT001 inhibited the expression of MYC with the IC50 value of 0.46 microM). FT001 has potent antiproliferative effects against MV-4-11 and demonstrates significant MYC mRNA suppression both in vitro and in vivo.
  • Shelf life instruction
    3 years
  • SMILES
    C(=O)(N1C=2C(N(C(C)=O)[C@@H](C)C1)=CC=C(C2)C3=CC=C(C=C3)N4CCS(=O)(=O)CC4)C5CC5
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200

References

  • Millan DS, et al. Design and Optimization of Benzopiperazines as Potent Inhibitors of BET Bromodomains. ACS Med Chem Lett. 2017 Jul 14;8(8):847-852.
    Read more