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GKI-1

HY-100521
MedChem Express
CAS Number2444764-03-6
Product group Chemicals
Estimated Purity99.89
Molecular Weight269.73
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Overview

  • Supplier
    MedChem Express
  • Product Name
    GKI-1 [2444764-03-6]
  • Delivery Days Customer
    9
  • CAS Number
    2444764-03-6
  • Estimated Purity
    99.89
  • Molecular Formula
    C15H12ClN3
  • Molecular Weight
    269.73
  • Scientific Description
    GKI-1 is a Greatwall (GWL) kinase inhibitor with IC 50 s of 4.9 and 2.5 microM against hGWL FL and hGWL-KinDom, respectively. GKI-1 robustly inhibits ROCK1 with an IC 50 of 11 microM, but only weakly affected PKA [1] .
  • SMILES
    ClC(C=C1)=CC=C1NC2=CC(C3=CNN=C3)=CC=C2
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200