Glucocorticoid receptor-IN-2 [2664932-65-2]

TargetMol Chemicals

Glucocorticoid receptor-IN-2 [2664932-65-2]

72

Chemical

Research Use Only

Glucocorticoid receptor-IN-2

C25H20F4N6O2

512.46

Glucocorticoid receptor-IN-2 is a selective regulator of the glucocorticoid receptor (GR) and exhibits anti-inflammatory activity. IC50: 0.171 nM) and also has some transcriptional activating effect on MMTV (EC50: 0.94 nM).

3 years

O([C@@H]([C@@H](NC(C(C)(F)F)=O)C)C1=CC(F)=CC(F)=C1)C=2C=C3C(N(N=C3)C4=CN5C(C=C4)=NN=C5)=CC2

-20°C

51202000