GP 1a [511532-96-0]

TargetMol Chemicals

GP 1a [511532-96-0]

4

511532-96-0

Chemical

Research Use Only

GP 1a

99.44%

C23H22Cl2N4O

441.35

GP 1a is a potent agonist of cannabinoid receptor 2 (CB2) (EC50=7.1), as shown in cAMP, GTPgammaS and beta-arrestin recruitment assays. GP 1a is approximately 30-fold more selective for CB2 receptors than CB1 receptors and increases P-ERK1/2 expression in HL-60 cells in vitro. GP 1a is beneficial for skin wound healing. GP 1a inhibits inflammation and fibrogenesis while promoting epithelial re-formation.

3 years

C(NN1CCCCC1)(=O)C=2C3=C(N(N2)C4=C(Cl)C=C(Cl)C=C4)C=5C(C3)=CC(C)=CC5

-20°C

12352200