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GR127935 (hydrochloride)

HY-100794
MedChem Express
CAS Number148642-42-6
Product group Chemicals
Estimated Purity99.38
Molecular Weight534.05
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Overview

  • Supplier
    MedChem Express
  • Product Name
    GR127935 (hydrochloride) [148642-42-6]
  • Delivery Days Customer
    10
  • CAS Number
    148642-42-6
  • Estimated Purity
    99.38
  • Molecular Formula
    C29H32ClN5O3
  • Molecular Weight
    534.05
  • Scientific Description
    GR127935 hydrochloride is a potent and orally active 5-HT1D and 5-HT1B receptor antagonist with pKis of 8.5 for both isoforms. GR127935 hydrochloride has 100-fold selectivity for 5-HT1B/1D receptors over 5-HT1A, 5-HT2A, and 5-HT2C receptors. GR127935 hydrochloride can be used in neurological disease research [1] [2] .
  • SMILES
    O=C(C1=CC=C(C2=CC=C(C3=NOC(C)=N3)C=C2C)C=C1)NC4=CC=C(OC)C(N5CCN(C)CC5)=C4.[H]Cl
  • Storage Instruction
    -20°C
  • UNSPSC
    12352200