GR127935 (hydrochloride)
HY-100794
Overview
- SupplierMedChem Express
- Product NameGR127935 (hydrochloride) [148642-42-6]
- Delivery Days Customer10
- CAS Number148642-42-6
- Estimated Purity99.38
- Molecular FormulaC29H32ClN5O3
- Molecular Weight534.05
- Scientific DescriptionGR127935 hydrochloride is a potent and orally active 5-HT1D and 5-HT1B receptor antagonist with pKis of 8.5 for both isoforms. GR127935 hydrochloride has 100-fold selectivity for 5-HT1B/1D receptors over 5-HT1A, 5-HT2A, and 5-HT2C receptors. GR127935 hydrochloride can be used in neurological disease research [1] [2] .
- SMILESO=C(C1=CC=C(C2=CC=C(C3=NOC(C)=N3)C=C2C)C=C1)NC4=CC=C(OC)C(N5CCN(C)CC5)=C4.[H]Cl
- Storage Instruction-20°C
- UNSPSC12352200