GRK5-IN-2

MedChem Express

GRK5-IN-2 [1642839-27-7]

10

1642839-27-7

Research Use Only

99.92

C20H20N4O4

380.40

GRK5-IN-2 (compound 707), a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor with an IC50 of 49.7 microM. GRK5-IN-2 regulates the expression and/or release of insulin and is useful for the metabolic disease research[1][2].

COC1=C(OC)C(OC)=CC(NC2=CC3=C(N=C(C4=CC=CO4)N3C)C=N2)=C1

-20°C,2°C to 8°C

12352200