GrTx1

MedChem Express

GrTx1

14

Research Use Only

C159H243N45O41S8

3697.43

GrTx1 is a peptide toxin originally isolated from the venom of the spider Grammostola rosea. GrTx1 blocks sodium channel, with IC50s of 0.63 microM, 0.23 microM, 0.77 microM, 1.29 microM, 0.63 microM and 0.37 microM for Nav1.1, Nav1.2, Nav1.3, Nav1.4, Nav1.6 and Nav1.7, repectively[2].GrTx1 can be used for neurological disease research[1].

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