GSK3368715 [1629013-22-4]

TargetMol Chemicals

GSK3368715 [1629013-22-4]

114

1629013-22-4

Chemical

Research Use Only

GSK3368715

C20H38N4O2

366.54

GSK3368715 is an orally active, reversible, and S-adenosyl-L-methionine (SAM) uncompetitive type I protein arginine methyltransferases (PRMTs) inhibitor (IC50s: 3.1 nM (PRMT1), 48 nM (PRMT3), 1148 nM (PRMT4), 5.7 nM (PRMT6), 1.7 nM (PRMT8)). It has strong anti-cancer activity.

3 years

C(OCC)C1(COCC)CCC(CC1)C=2C(CN(CCNC)C)=CNN2

-20°C

12352200