GSK494581A

MedChem Express

GSK494581A

9

Research Use Only

C27H28F2N2O4S

514.58

GSK494581A is a specific ligand for human GPR55 (pEC 50 of 6.8) and also acts as an inhibitor of glycine transporter subtype 1 ( GlyT1 ). GSK494581A may regulate pain signaling, bone morphogenesis, and vascular endothelial cell formation by binding to GPR55 [1] .

O=C(N1CCN(C2=CC=C(C(OC)C)C=C2F)CC1)C3=CC(S(=O)(C)=O)=CC=C3C4=CC=C(F)C=C4

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