GSK931145

MedChem Express

GSK931145

9

Research Use Only

C23H30N2O

350.50

GSK931145 is a glycine transporter 1 (GlyT1) inhibitor with anti-epileptic activity. GSK931145 exhibits a low minimum effective dose in the maximum electrical stimulation threshold test, indicating that it has a significant anti-epileptic effect. GSK931145 is also suitable as a positron emission tomography (PET) radioligand for quantifying the availability of glycine transporters in the living brain [1] .

O=C(C1=C(C)C=CC=C1C)NC(C2(CCCC2)N(C)C)C3=CC=CC=C3

12352200