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GYKI-47261 dihydrochloride

T38601
TargetMol Chemicals
CAS Number1217049-32-5
Product group Chemicals
Molecular Weight395.71
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    GYKI-47261 dihydrochloride
  • Delivery Days Customer
    1001
  • CAS Number
    1217049-32-5
  • Category Supplier
    Chemical
  • Chemical Name
    GYKI-47261 dihydrochloride
  • Molecular Formula
    C18H17Cl3N4
  • Molecular Weight
    395.71
  • Scientific Description
    GYKI-47261 dihydrochloride is a selective AMPA receptor antagonist, administered orally, and exhibits competitive activity with an IC 50 of 2.5 uM. It displays a wide range of anticonvulsive effects and demonstrates neuroprotective properties. Additionally, GYKI-47261 dihydrochloride is a potent inducer of CYP2E1.
  • Shelf life instruction
    3 years
  • SMILES
    Cl.Cl.Cc1cn2N=C(c3ccc(N)cc3)c3cc(Cl)ccc3Cc2n1 ;t:4;
  • Storage Instruction
    -20°
  • UNSPSC
    12352200

References

  • Tamási V, et al. GYKI-47261, a new AMPA [2-amino-3-(3-hydroxymethylisoxazole-4-yl)propionic acid] antagonist, is a CYP2E1 inducer. Drug Metab Dispos. 2003;31(11):1310-1314.