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IACS-9571

IACS-9571

T11597
TargetMol Chemicals
CAS Number1800477-30-8
Product group Chemicals
Molecular Weight642.76
Price on request
Packing Size
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Overview

  • Supplier
    TargetMol Chemicals
  • Product Name
    IACS-9571
  • Delivery Days Customer
    65
  • CAS Number
    1800477-30-8
  • Category Supplier
    Chemical
  • Chemical Name
    IACS-9571
  • Molecular Formula
    C32H42N4O8S
  • Molecular Weight
    642.76
  • Scientific Description
    IACS-9571 is a selective and potent inhibitor of TRIM24 and BRPF1, (IC50: 8 nM for TRIM24; Kds: 31 nM and 14 nM for TRIM24 and BRPF1).
  • Shelf life instruction
    3 years
  • SMILES
    CN1C=2C(=CC(NS(=O)(=O)C3=CC(OC)=C(OC)C=C3)=C(OC4=CC(OCCCCN(C)C)=CC(OCCC)=C4)C2)N(C)C1=O
  • Storage Instruction
    -20°
  • UNSPSC
    12352200

References

  • Palmer WS, et al. Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor. J Med Chem. 2016 Feb 25;59(4):1440-54.
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