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Irdabisant (hydrochloride)

HY-109968A
MedChem Express
Molecular Weight349.86
Product group Chemicals
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Overview

  • Supplier
    MedChem Express
  • Product Name
    Irdabisant (hydrochloride)
  • Delivery Days Customer
    10
  • Certification
    Research Use Only
  • Molecular Formula
    C18H24ClN3O2
  • Molecular Weight
    349.86
  • Scientific Description
    Irdabisant (CEP-26401) hydrochloride is a selective, orally active and blood-brain barrier (BBB) penetrant histamine H3 receptor (H3R) inverse agonist/inverse agonist with K i values of 7.2 nM and 2.0 nM for rat H3R and human H3R, respectively. Irdabisant hydrochloride has relatively low inhibitory activity against hERG current with an IC 50 of 13.8 microM. Irdabisant hydrochloride has cognition-enhancing and wake-promoting activities in the rat social recognition model. Irdabisant hydrochloride can be used to research schizophrenia or cognitive impairment [1] [2] .
  • SMILES
    C[C@H](CCC1)N1CCCOC2=CC=C(C(C=C3)=NNC3=O)C=C2.[H]Cl
  • UNSPSC
    12352200