KDM1/CDK1-IN-1
HY-147901
Molecular Weight431.47
Product group Chemicals
Overview
- SupplierMedChem Express
- Product NameKDM1/CDK1-IN-1
- Delivery Days Customer10
- CertificationResearch Use Only
- Molecular FormulaC22H17N5O3S
- Molecular Weight431.47
- Scientific DescriptionKDM1/CDK1-IN-1 (compound 4) is a potent KDM1 and CDK1 inhibitor, with IC50 values of 0.096 and 0.078 microM, respectively.KDM1/CDK1-IN-1 induces cell cycle arrest at G2/M phase and apoptosis in HOP-92 cells. KDM1/CDK1-IN-1 exhibits potent cytotoxic activity against the CCRF-CEM, HOP-92 and Hep-G2 cells, with IC50 values of 16.34, 3.45 and 7.79 microM, respectively.
- SMILESO=C(C1=C(O)N2C(N=C1)=C(C3=NC4=CC=CC=C4S3)C(NC5=CC=CC=C5)=N2)OCC
- Storage InstructionSee Manual
- UNSPSC12352200