Bio-Connect

Leucettinib-92 [2732859-57-1]

HY-155723
MedChem Express
CAS Number2732859-57-1
Product group Chemicals
Estimated Purity98.54
Molecular Weight378.49
Sign in to order and to see your custom pricing.
Large volume orders?
Order with a bulk request

Overview

  • Supplier
    MedChem Express
  • Product Name
    Leucettinib-92 [2732859-57-1]
  • Delivery Days Customer
    14
  • CAS Number
    2732859-57-1
  • Certification
    Research Use Only
  • Estimated Purity
    98.54
  • Molecular Formula
    C21H22N4OS
  • Molecular Weight
    378.49
  • Scientific Description
    Leucettinib-92 (compound 92) is an inhibitor of DYRK/CLK kinase, The IC50s are 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 microM (CLK3), 124 nM (DYRK1A), 204 nM (DYRK1B), 0.16 microM (DYRK2), respectively. 1.0 microM (DYRK3), 0.52 microM (DYRK4), 2.78 microM (GSK3)[1].
  • SMILES
    O=C(N1)/C(N=C1NC2(C3)C[C@H]4C[C@@H]3C[C@@H](C2)C4)=C/C5=CC=C(N=CS6)C6=C5
  • Storage Instruction
    2°C to 8°C
  • UNSPSC
    12352200