Linaprazan (mesylate)

MedChem Express

Linaprazan (mesylate)

9

C22H30N4O5S

462.56

Linaprazan mesylate can inhibit H+,K+ -ATPase in the stomach through K+ competitive binding. (IC 50: 1.0 +/- 0.2 microM), it has a strong inhibitory effect on acid. Linaprazan (AZD0865) mesylate can be used for research on reflux esophagitis with oral activity [1] [2] [3] .

O=C(C1=CN2C(C(NCC3=C(C)C=CC=C3C)=C1)=NC(C)=C2C)NCCO.CS(=O)(O)=O

12352200