Lintitript

MedChem Express

Lintitript [136381-85-6]

9

136381-85-6

Research Use Only

99.58

C20H14ClN3O3S

411.86

Lintitript (SR 27897) is a highly potent, selective, orally active, competitive and non-peptide cholecystokinin (CCK1) receptor antagonist with an EC 50 of 6 nM and a K i of 0.2 nM. Lintitript displays > 33-fold selectivity more selective for CCK1 than CCK2 receptors ( EC 50 value of 200 nM). Lintitript increases plasma concentration of leptin and food intake as well as plasma concentration of insulin [1] [2] [3] .

O=C(O)CN1C(C(NC2=NC(C3=CC=CC=C3Cl)=CS2)=O)=CC4=C1C=CC=C4

-20°C,2°C to 8°C

12352200