MCHR1 antagonist 4 [1574538-43-4]

TargetMol Chemicals

MCHR1 antagonist 4 [1574538-43-4]

9

Research Use Only

C26H30N2O4

434.53

MCHR1antagonist 4 (Compound 2m) is an MCHR1 antagonist capable of penetrating the blood-brain barrier, with Ki values of 0.74 nM and 0.76 nM for hMCHR1 and rMCHR1, respectively. Additionally, it serves as an effective anti-obesity agent.

O=C1C(OC2=CC=C(C=C2)C3CC3)=CCN1C4=CC=C(OCCN5CCCC5)C(OC)=C4

-20°C

12352200