MM-589 (racemic mixture ) (TFA)
HY-100869B
Overview
- SupplierMedChem Express
- Product NameMM-589 (racemic mixture ) (TFA)
- Delivery Days Customer14
- Estimated Purity99.83
- Molecular FormulaC30H45F3N8O7
- Molecular Weight686.72
- Scientific DescriptionMM-589 (racemic mixture) TFA, is a racemic mixture of MM-589 TFA (HY-100869A). MM-589 TFA is a potent inhibitor of WD repeat domain 5 (WDR5) and mixed lineage leukemia (MLL) protein-protein interaction. MM-589 binds to WDR5 with an IC 50 of 0.90 nM and inhibits the MLL H3K4 methyltransferase activity with an IC 50 of 12.7 nM [1] .
- SMILESO=C(NCC[C@](NC(C(C)C)=O)(C)C1=O)[C@H](NC([C@@H](NC([C@H](CCCNC(NC)=N)N1)=O)CC)=O)C2=CC=CC=C2.O=C(NCC[C@](NC(C(C)C)=O)(C)C3=O)[C@@H](NC([C@@H](NC([C@H](CCCNC(NC)=N)N3)=O)CC)=O)C4=CC=CC=C4.OC(C(F)(F)F)=O.[(7:3)]
- Storage Instruction-20°C
- UNSPSC12352200