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Mozavaptan

M1917
AbMole BioScience
CAS Number137975-06-5
Product group Chemicals
Estimated Purity0.9912
Molecular Weight427.53
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Overview

  • Supplier
    AbMole BioScience
  • Product Name
    Mozavaptan
  • Delivery Days Customer
    9
  • CAS Number
    137975-06-5
  • Category Supplier
    Chemical
  • Certification
    Research Use Only
  • Estimated Purity
    0.9912
  • Molecular Formula
    C27H29N3O2
  • Molecular Weight
    427.53
  • Scientific Description
    Mozavaptan (OPC-31260) is a benzazepine derivative and a potent, selective, competitive and orally active vasopressin V2 receptor antagonist with an IC50 of 14 nM. Mozavaptan shows ~85-fold selectivity for V2 receptor over V1 receptor (IC50 of 1.2 uM), and can antagonize the antidiuretic action of arginine vasopressin (AVP) in vivo.
  • SMILES
    CN(C)C1CCCN(C(=O)C2=CC=C(NC(=O)C3=C(C)C=CC=C3)C=C2)C4=C1C=CC=C4
  • UNSPSC
    12352200