MRS2179 (tetrasodium)

MedChem Express

MRS2179 (tetrasodium) [1454889-37-2]

10

1454889-37-2

Research Use Only

C11H13N5Na4O9P2

513.16

MRS2179 tetrasodium is a competitive P2Y1 receptor antagonist, with a K b of 102 nM and a pA 2 of 6.99 for turkey P2Y1 receptor. MRS2179 tetrasodium is selective for P2Y1 over P2X1 (IC 50 =1.15 microM), P2X3 (12.9 microM), P2X2, P2X4, P2Y2, P2Y4, and P2Y6 receptors [1] [2] . MRS2179 tetrasodium inhibits platelet aggregation [3] .

CNC1=C2C(N([C@](C[C@@H]3O[P](O[Na])(O[Na])=O)([H])O[C@@H]3CO[P](O[Na])(O[Na])=O)C=N2)=NC=N1

12352200