MRS2179 (tetrasodium hydrate)

MedChem Express

MRS2179 (tetrasodium hydrate)

10

99.6

C11H13N5O9P2Na4.31/2H2O

576.21

MRS2179 tetrasodium hydrate is a competitive P2Y1 receptor antagonist, with a K b of 102 nM and a pA 2 of 6.99 for turkey P2Y1 receptor. MRS2179 tetrasodium hydrate is selective for P2Y1 over P2X1 (IC 50 =1.15 microM), P2X3 (12.9 microM), P2X2, P2X4, P2Y2, P2Y4, and P2Y6 receptors [1] [2] . MRS2179 tetrasodium hydrate inhibits platelet aggregation [3] .

CNC1=C2C(N([C@](C[C@@H]3O[P](O[Na])(O[Na])=O)([H])O[C@@H]3CO[P](O[Na])(O[Na])=O)C=N2)=NC=N1.O.[3.5]

-20°C

12352200