MRS2365

MedChem Express

MRS2365

10

Research Use Only

C13H19N5O9P2S

483.33

MRS2365 is a potent and selective P2Y1 receptor ( EC 50 =0.4 nM) / [ 35 S]GTPgammaS binding/ beta-arrestin 2 recruitment agonist with an EC 50 of 0.4 nM. MRS2365 relieves mechanical allodynia and increases mechanical sensitivity. MRS2365 shows little agonist or antagonist activity at the P2Y12 or P2Y13 receptors [1] [2] [3] [4] .

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